Skip to main content
PepStack

Cortisol

Adrenal Hormones
HydrocortisoneCompound FCortef

Overview

Cortisol, also known as hydrocortisone, Compound F, or Cortef, is an endogenous glucocorticoid hormone produced by the adrenal cortex. It belongs to the steroid hormone class and plays a crucial role in various physiological processes. Cortisol is synthesized from cholesterol and is released in response to stress and low blood-glucose concentration. Synthetic forms of cortisol are used in medicine to treat a variety of conditions. Researchers have extensively studied cortisol due to its significant impact on the body's stress response and metabolic functions. It is primarily involved in the regulation of metabolism, immune response, and maintenance of homeostasis. Cortisol's role in the body's response to stress, inflammation, and circadian rhythms has been a major focus of research. Its dysregulation is associated with conditions such as Cushing's syndrome and Addison's disease. Cortisol exerts its effects by binding to glucocorticoid receptors, which are part of the nuclear receptor superfamily. Upon binding, the hormone-receptor complex translocates to the nucleus, where it influences the transcription of target genes involved in glucose metabolism, immune response, and other vital processes. Researchers have found that cortisol's action involves complex signaling pathways that modulate various physiological responses. The pharmacokinetic properties of cortisol include a circulating half-life of approximately 70 minutes. It is metabolized primarily in the liver and excreted in urine. Oral bioavailability is limited due to first-pass metabolism. Cortisol is used clinically in its synthetic form to treat inflammatory and autoimmune conditions, among others. It is approved by regulatory agencies like the FDA for various therapeutic uses. Researchers have observed its efficacy in managing conditions such as asthma, rheumatoid arthritis, and adrenal insufficiency. Its use is regulated and requires a prescription.

Mechanism of Action

Cortisol acts primarily on glucocorticoid receptors, which are intracellular receptors that, upon activation, translocate to the cell nucleus. This activation leads to the modulation of gene expression, affecting processes such as glucose metabolism, immune response, and inflammation control.

Molecular Data

FormulaC21H30O5
Molecular Weight362.5 g/mol
CAS Number50-23-7
PubChem CID5754

Half-Life & Pharmacokinetics

EndogenousCirculating half-life ~70 minutes
Intravenous~10 minutes
OralPoor bioavailability due to first-pass metabolism

Synthetic forms may have different pharmacokinetic profiles depending on formulation.

Storage

Temperature

Store at room temperature (15-30°C)

Light

Protect from light

Form

Aqueous solution: use within specified time after opening

Notes

Ensure container is tightly closed to prevent contamination.

Solubility

Cortisol is poorly soluble in water but soluble in ethanol and other organic solvents.

Legal Status

🇩🇪DE

Prescription only (verschreibungspflichtig), not a controlled substance under BtMG.

🇺🇸US

FDA approved for medical use, prescription required.

🇦🇺AU

TGA Schedule 4 (S4), prescription only.

🇬🇧UK

Prescription only medicine (POM) under MHRA regulations.

Legal status information is provided for general reference only and may not reflect the most current regulatory changes. Always verify with official government sources before making any decisions.

7 Research Publications

Hippocampal Mechanisms Support Cortisol-Induced Memory Enhancements.

Human

The Journal of neuroscience : the official journal of the Society for Neuroscience · 2023

Researchers found that cortisol, a stress hormone, can enhance the memory of emotionally significant information. They observed that cortisol improved the brain's connectivity in the hippocampus, which is crucial for forming memories, leading to better recall of positive experiences.

  • Cortisol enhances the encoding of emotionally charged memories.
  • Increased connectivity in the hippocampus is linked to better memory performance under cortisol.
  • The way the hippocampus processes memories changes when cortisol is present.
PubMed

Prophylactic postnatal corticosteroids: Early hydrocortisone.

Review

Seminars in fetal & neonatal medicine · 2019

Researchers found that giving low-dose hydrocortisone to extremely preterm infants can significantly reduce the risk of bronchopulmonary dysplasia (BPD) and improve survival rates. They observed that this treatment did not lead to increased gastrointestinal issues or negatively affect long-term development, despite a slight rise in late-onset infections in the most vulnerable infants.

  • Low-dose hydrocortisone reduced the incidence of BPD and mortality in preterm infants.
  • There was no increase in gastrointestinal perforation without indomethacin treatment.
  • Late-onset sepsis increased in the most immature infants but did not affect overall survival or development.
PubMed

Human studies on hypothalamo-pituitary-adrenal (HPA) axis.

Review

Best practice & research. Clinical endocrinology & metabolism · 2017

Researchers observed that the body's daily rhythm of cortisol, a stress hormone, is influenced by the brain's central clock. Changes in this rhythm, often seen in shift workers and certain health conditions, can lead to serious health issues, including metabolic problems and increased risk of depression. Efforts to improve cortisol replacement therapies aim to restore this rhythm and enhance patients' quality of life.

  • Shift work and certain health conditions disrupt the normal cortisol rhythm.
  • Higher cortisol levels are linked to serious health risks, including metabolic issues.
  • New therapies aim to better mimic the natural cortisol rhythm to improve patient outcomes.
PubMed

Salivary cortisol and cortisone in the clinical setting.

Review

Current opinion in endocrinology, diabetes, and obesity · 2017

Researchers found that measuring cortisol and cortisone in saliva can effectively assess adrenal function and diagnose conditions related to hormone imbalance. They observed that salivary cortisone is particularly useful when serum cortisol levels are low or when patients are on hydrocortisone therapy, as it provides more accurate results without contamination issues.

  • Salivary measurements detect only free hormones and can be taken easily during daily routines.
  • Salivary cortisone is a better marker than salivary cortisol for low serum cortisol levels.
  • Salivary biomarkers are more accurate for assessing adrenal reserve compared to serum cortisol.
PubMed

Is physiological glucocorticoid replacement important in children?

Review

Archives of disease in childhood · 2017

Researchers observed that children with adrenal insufficiency often experience fatigue and poor quality of life due to unbalanced cortisol levels from current treatments. They highlighted the potential benefits of new therapies that more closely mimic the body's natural cortisol rhythm, which could improve health outcomes for these patients.

  • Current glucocorticoid treatments lead to unphysiological cortisol levels.
  • Patients report fatigue and poor quality of life.
  • New therapies may better replicate natural cortisol patterns.
PubMed

Recent Advances in Hydrocortisone Replacement Treatment.

Review

Endocrine development · 2016

Researchers observed that traditional hydrocortisone treatments for cortisol deficiency do not mimic the body's natural rhythm, which may lead to health issues. Recent advancements, including modified-release formulations and continuous infusions, show promise in improving treatment outcomes. Larger studies are needed to confirm these benefits for patients.

  • Conventional hydrocortisone treatment is inadequate and does not replicate natural cortisol rhythms.
  • New treatment methods have shown clinical and biochemical improvements in initial studies.
  • Further research is required to assess long-term benefits of these innovative approaches.
PubMed

Compound f: the history of hydrocortisone and hand surgery.

Human

The Journal of hand surgery · 2013

Researchers observed the significant history of hydrocortisone, a medication widely used in hand surgery for treating various orthopedic conditions. They highlighted the collaboration between physicians and researchers that led to its discovery and clinical application, emphasizing the focus on patient care at Mayo Clinic.

  • Hydrocortisone is effective for treating conditions like tendinitis and carpal tunnel syndrome.
  • The development of cortisone and hydrocortisone was influenced by collaborative research efforts.
  • The history of these medications underscores the commitment to patient care in medical practice.
PubMed

Track your hormone research in PepStack

Log cycles, set reminders and visualize serum levels.

This page is for informational and research purposes only. All information is based on published scientific literature. Nothing on this page constitutes medical advice or replaces consultation with a qualified healthcare professional.