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DHEA-S

Adrenal Hormones
DHEASDehydroepiandrosterone sulfate

Overview

Dehydroepiandrosterone sulfate (DHEA-S) is an endogenous steroid hormone primarily produced by the adrenal glands, with minor contributions from the gonads and brain. It belongs to the class of adrenal hormones and is a sulfated form of dehydroepiandrosterone (DHEA), which is a precursor to androgens and estrogens. DHEA-S is one of the most abundant circulating steroids in humans and serves as a reservoir that can be converted into more active steroid hormones. Researchers have found that DHEA-S plays a role in various physiological processes, including immune function, metabolism, and the development of secondary sexual characteristics. It is also a subject of interest in research areas such as aging, cardiovascular health, and neuroprotection. The mechanism of action of DHEA-S involves its conversion to DHEA, which then interacts with androgen and estrogen receptors, influencing a wide range of biological pathways. Researchers have observed that these pathways can affect cellular proliferation, differentiation, and apoptosis. DHEA-S itself does not directly bind to these receptors but serves as a precursor. Pharmacokinetically, DHEA-S has a relatively long circulating half-life of approximately 7 to 10 hours, allowing it to maintain stable levels in the bloodstream. It is metabolized primarily in the liver and excreted in urine. Oral bioavailability is limited due to first-pass metabolism. Clinically, DHEA-S levels are measured to assess adrenal function and diagnose disorders such as adrenal insufficiency or hyperplasia. It is not approved as a therapeutic agent in many countries, and its use is primarily limited to research settings. Regulatory standing varies, with some regions allowing over-the-counter sales of DHEA supplements, which can affect DHEA-S levels indirectly.

Mechanism of Action

DHEA-S acts primarily as a precursor to DHEA, which then interacts with androgen and estrogen receptors. This conversion facilitates biological cascades that influence cellular processes such as proliferation and differentiation, impacting various physiological functions.

Molecular Data

FormulaC19H28O5S
Molecular Weight368.5 g/mol
CAS Number651-48-9
PubChem CID12594

Half-Life & Pharmacokinetics

EndogenousCirculating half-life ~7 to 10 hours
OralPoor bioavailability due to first-pass metabolism

DHEA-S is primarily measured in its endogenous form; synthetic administration is uncommon.

Storage

Temperature

Store at room temperature (15-30°C)

Light

Protect from light

Form

Stable in solid form for extended periods

Notes

Ensure container is tightly sealed to prevent moisture absorption.

Solubility

DHEA-S is water-soluble due to its sulfate group, facilitating its circulation in the bloodstream.

Legal Status

🇩🇪DE

DHEA-S is not a controlled substance but may require a prescription for therapeutic use.

🇺🇸US

DHEA is available as an over-the-counter supplement; DHEA-S itself is not FDA-approved as a drug.

🇦🇺AU

DHEA is classified as a Schedule 4 (S4) substance, requiring a prescription.

🇬🇧UK

DHEA-S is not classified as a prescription-only medicine (POM) but is not widely available as a therapeutic agent.

Legal status information is provided for general reference only and may not reflect the most current regulatory changes. Always verify with official government sources before making any decisions.

8 Research Publications

Aging induces region-specific dysregulation of hormone synthesis in the primate adrenal gland.

Unknown

Nature aging · 2024

Researchers found that aging affects hormone production in the adrenal glands, which are important for metabolism and stress responses. They observed that specific areas of the adrenal glands showed significant changes in hormone synthesis and cell function as primates aged, indicating potential targets for improving health in older adults.

  • Aging disrupts lipid metabolism and hormone production in the adrenal glands.
  • The zona reticularis region, responsible for producing a key hormone, is particularly affected by aging.
  • Reduced cholesterol uptake in adrenal cells may contribute to age-related hormone deficiencies.
PubMed

Correlation between salivary dehydroepiandrosterone sulfate (DHEA-S) levels and cervical vertebral maturation in Saudi individuals.

Review

The Saudi dental journal · 2022

Researchers observed a link between levels of a hormone called DHEA-S in saliva and the growth stages of cervical vertebrae in young people. This suggests that measuring DHEA-S could help identify when a person is experiencing a growth spurt during puberty, offering a non-invasive way to track development.

  • DHEA-S levels varied significantly at specific cervical maturation stages.
  • Higher DHEA-S levels were associated with advanced growth stages.
  • Salivary DHEA-S may serve as a useful indicator of pubertal growth.
PubMed

Steroid Sulfation in Adrenal Tumors.

Review

The Journal of clinical endocrinology and metabolism · 2021

Researchers observed that steroid sulfates, particularly dehydroepiandrosterone sulfate (DHEAS), play a significant role in adrenal tumors and may serve as useful biomarkers for diagnosis. They highlighted that recent advancements in analytical techniques could enhance the study of these sulfated steroids, which have important biological functions beyond their traditional roles.

  • Steroid sulfates are linked to the development of adrenal tumors.
  • DHEAS levels may help in diagnosing certain adrenal conditions.
  • New analytical methods can improve the understanding of steroid sulfation in adrenal health.
PubMed

Dehydroepiandrosterone (DHEA) and Its Sulfate (DHEA-S) in Mammalian Reproduction: Known Roles and Novel Paradigms.

Review

Vitamins and hormones · 2018

Researchers observed that dehydroepiandrosterone (DHEA) plays a crucial role in mammalian reproduction by serving as a precursor for important sex hormones. They found that DHEA supplementation may help improve ovarian function and that steroid hormones like estradiol and testosterone are essential for the maturation of eggs in the ovaries.

  • DHEA is a key precursor for sex hormones in mammals.
  • DHEA supplementation may enhance ovarian reserve.
  • Steroid hormones are important for the maturation of eggs.
PubMed

Dehydroepiandrosterone and Dehydroepiandrosterone-Sulfate and Emotional Processing.

Unknown

Vitamins and hormones · 2018

Researchers found that the steroid hormones dehydroepiandrosterone (DHEA) and its sulfate form (DHEAS) may influence how we process emotions. Higher levels of these hormones are linked to reduced activity in brain areas associated with negative emotions, potentially protecting against depression while enhancing attention and memory.

  • Higher DHEA(S) levels may reduce negative emotional processing.
  • DHEA(S) is associated with better attention and working memory.
  • DHEA(S) may protect against negative emotions and depression.
PubMed

Dehydroepiandrosterone sulfate (DHEAS) as an endocrine marker of aging in calorie restriction studies.

Review

Experimental gerontology · 2013

Researchers found that dehydroepiandrosterone sulfate (DHEAS), a hormone often linked to aging, decreases as animals age. However, in studies where calorie intake was reduced, this decline in DHEAS levels was not significantly prevented, suggesting that dietary changes might affect how this hormone is processed in the body. This raises questions about the reliability of DHEAS as a marker of aging in calorie restriction studies.

  • DHEAS levels are high in young adulthood and decline with age.
  • Caloric restriction did not prevent the decline of DHEAS in old rhesus macaques.
  • Dietary changes may alter the metabolism of DHEAS, affecting its reliability as an aging marker.
PubMed

DHEA and DHEA-S: a review.

Review

Journal of clinical pharmacology · 1999

Researchers observed that DHEA and its related hormone DHEA-S are produced by the adrenal glands and play a role in various bodily functions. The review highlights how levels of these hormones can change with age, gender, health conditions, diet, and exercise, as well as the effects of certain medications. The article also discusses their potential links to stress, brain function, immune response, and heart health.

  • DHEA and DHEA-S levels vary with age and gender.
  • Hormone concentrations are influenced by diet, exercise, and medications.
  • DHEA and DHEA-S may be related to stress, brain health, immune function, and cardiovascular issues.
PubMed

Dehydroepiandrosterone metabolism.

Review

The Journal of endocrinology · 1996

Researchers observed that dehydroepiandrosterone (DHEA) and its sulfate form (DHEAS) are found in the blood, with DHEA being cleared quickly while DHEAS takes longer. They also found that these two forms can convert into each other and are important for producing hormones like testosterone and estrogen in the body.

  • DHEA is cleared from the blood rapidly, while DHEAS is cleared more slowly.
  • About 6% of DHEA converts back into DHEAS, while 60-70% of DHEAS converts back into DHEA.
  • Both DHEA and DHEAS can be converted into other hormones, including testosterone and estrogen.
PubMed

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This page is for informational and research purposes only. All information is based on published scientific literature. Nothing on this page constitutes medical advice or replaces consultation with a qualified healthcare professional.